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LIMU 2nd

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All the following side effect of 1st generation except:Anonymous voting
  • Sedation.
  • Atropine like action
  • Orthostatic hypotension
  • Ventricular arrhythmia
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regarding the 1st generation of H1-R blocker drugs all of the following is true exceptAnonymous voting
  • Highly lipid solubel,crossBBB.
  • Short duration of action.
  • More potent than 2nd generation.
  • Cheap.
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๐ŸŸก ู…ุนู„ูˆู…ุฉ ู†ุจู‡ุช ุนู„ูŠู‡ุง ุงู„ุฏูƒุชูˆุฑุฉ ู‚ุฏ ุชุฃุชูŠ ูƒุณุคุงู„: Doctor prescribe 1st generation anti histamine for patient, the patient should be avoid:Anonymous voting
  • Eating fried chicken.
  • Watching movies.
  • Driving a car.
  • Setting in the garden.
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ู‡ุฐูŠู† ูƒู„ ูˆุฃู‡ู… ู…ูˆุงุถูŠุน ุงู„Histamine.
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๐ŸŸกAll H2 blocker end by suffix (tidine). ุฃู‡ู…ู‡ู† cimitidine.
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๐ŸŸกCyproheptadine. ุงู„ุฏูˆุงุก ููŠู‡ ุงุณู… ู‡ุจุฉ ูˆุงู„ุฐูŠ ูŠุนู†ูŠ ู‡ุฏูŠุฉ. ู‡ุฏูŠุฉ histamine 1R blcck . ุจุนุฏู‡ุง ุถุญูƒ (serotonin (5HT2R block. H1blocker. 5HT2R blocker. ๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡๐Ÿ‘‡
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๐ŸŸกpromethazine ู„ู‡ ู…ูŠุฒุชูŠู†ร—2 H1 blocker alpha1 blocker=>orthostatic hypotension ................. and close Na channel so can use as local anesthesia.
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๐ŸŸก1st generation of H1 blocker ุงู„ุดูŠุฎ ู…ู† ุงู„ุทุฑุงุฒ ุงู„ู‚ุฏูŠู…. ุชุฃุซูŠุฑ ุถุนูŠู ูˆู„ูˆู‚ุช ู‚ุตูŠุฑ ูˆุฏุงุฆู…ุง ุตุงุญุจ ุญูƒู…ุฉ(,lipid soluble cross BBB). ุณุคุงู„ ู…ู‡ู… ูˆู…ุถู…ูˆู† ูˆู„ุง ูŠุฎู„ูˆ ู…ู†ู‡ ุงู…ุชุญุงู†.
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